Computer-Aided Drug Design

Drug Design Projects in Progress

CollaboratorInstitutionTarget/Status
Archontis & SpirosUniv. of Cyprusglycogen phosphorylase, lead optimization in progress
CoopUMB, PharmacyOpioids/Analgesics, lead optimization in progress, NIH R01; funded
DiGateUMB, PharmacyTopoisomersase, active cmp identified NIH R21; submitted
HayashiUMB, Pharmacyp56lck kinase, active cmpds identified, patent pend. NIH R01; funded
NeamatiUSC, PharmacyHIV Integrase, active cmpd identified, publications, NIH R01; submitted
OikonomakosInst. Organic & Pharmaceutical Chem. Nat. Hellenic Res. Fd. Greeceglycogen phosphorylase/phosphorylase kinase, Greek Secretariat for Research and Technology, International S & T Cooperation Directorate, Grant; submitted
Passaniti

UMB, Medicine

Runt Domain/angiogenesis, active cmpds identified, NIH R21; funded
SerreroUMB, PharmacyPCDGF/breast cancer, active cmpds identified, DoD Concept Award; Funded
ShapiroUMB, PharmacyERK kinase, active cmpds identified, NIH R21; funded
SrivistavaUMB, Pharmacy

Death Receptor/Apoptosis, CADD screen complete, DoD Idea Award; Funded

SussmanUMB, Pharmacyb-Catenin/colon Cancer, active cmpds identified, NIH R21; funded
WeberUMB, MedicineS100b - P53 Interactions, Active cmpds identified, ACS funded, NIH R01; submitted
ZhangUniv. of Texas, Southwest Med. CenterAdenosyltransferase, Active compounds identified. NIH R01 submitted.